Intermediates
Class Product
   
Antibiotic: β - Lactamic Intermediates 3- TZ
  6-APA
  7-ACA
  7-HACA (7-ACA Desacetyl)
  7-ACT
  7-ADCA
  7-AVNA
  7-PACA (or 7- ARPA)
  7-TDCA
  Penicillin G Potassium Crude
Ciprofloxacin & Enrofloxacin Q-Acid 
Cephalosporin Intermediates 7-ACCA 
  7-ANCA 
  7-AMCA 
  7-APRA 
  7-AVCA
Anastrazole & int 2-[3-(Cyano-dimethyl-methyl)-5-methyl-phenyl]-2-methyl-propionitrile 
Amisulpride and int. 2-methoxy-4-amino-5-ethyl sulfonyl benzoic acid
Atorvastatin & ATS-5 ATS-8 ATS -9 M 4 L 1 ATS-5 : (R)-4-cyano-3-hydroxybutyric acid ethyl ester
  ATS-8 : (4R,Cis)-1,1-dimethylethyl-cyanomethyl-2,2- dimethyl-1,3-dioxane-4-acetate
Atovaquone Trans-4-chlorophenyl-1-cyclohexane carboxylicacid
4-AA (3s,4r)-4-acetoxy-3-[(r)-1-(tert-butyldimethylsilyloxy)ethyl]azetidin-2-1
Bicalutamide and int N-[4-Cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorophenyl)thio]-2-hydroxy-2-methylpropionamide
Candesartan Cilexetil  N-( Triphenylmethyl) ¨C 5-( 4'-bromomethylbiphenyl-2yl) tetrazole
Cilostazole  5-(4-Chlorobutyl)-1-Cyclohexyl-1H-Tetrazole
  6-Hydroxy-3,4-dihydro-2(1H)-quinolinone
Clopidogrel  2-Thiophene Ethanol 
  (+)-Methyl-alpha-(2-Thienylethamino) (2-Chlorophenyl) AcetateHydrochloride 
  N-[(2-Thienyl)ethyl]-(2s)-2-chloro-phenyl Glycine methyl ester 
Cyproterone Acetate 1, 2a -Methylene-6-didehydro -17a -acetoxy Progesterone
  1-Chloromethyl-6-chloro-6-dehydro -17a -acetoxy Progesterone
CPP 2,3-cyclopenteno pyridine
Donepezil  5,6-Dimethoxy-1-Indanone 
  N-Benzyl Piperidine-4-Carboxaldehyde 
Doxofylline and Int. 2-Bromethyl 1,3 dioxolane
EHATA Ethyl(Z)-2-(2-Aminothiazole-4-yl)-2-Methoxyimino Acetate
Exemestane Androsta-1,4-dien-3-one,17-hydoxy-6-methylene(17,β)
  Androsta-4-ene-3,17-dione,6-methylene(17,β)
Faropenem and Int Ally(1R,2R,5R,6S)-6(1-tert-butyldimethyl siloxyethyl)-2
Gemcitabine &int 2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate
  2-Deoxy-2,2-difluoro pentofuranos-1-ulose-3,5-dibenzoate
  2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dicinnamate-1-methane sulfonate
  2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dicinnamate
Ibandronate Sodium 3-(N-methylpentylamino)propionic acid hydrochloride
Imiquimod and int N4-(2-Methylpropyl-3,4-Quinolinediamin
Montelukast sodium 1-(1-(s)-(3-(2-(7-chloro-2-qionolinyl)-ethenyl-phenyl)-3-hydroxy-propyl)phenyl)-2-propanol
MICA ACID (Z)-2-(tert-methoxycarbonyl methoxyimino)-2-(2-aminothiazol-4-yl) acetic acid
MICA ESTER S-2-benzothiazolyl (Z)-2-(2-aminothiazol-4-yl)-2-methoxycarbonylmethoxyiminothio acetate
Olanzapine  4-Amino-2-Methyl-10H-Thieno[2,3-b][1,5]Benxodiazepine Hcl 
Olmesartan & int 4-chloromethyl-5-methyl-1,3-Dioxol-2-one (DMDO-CL)
  Trityl Olmesartan Medoxomil
Olopatadine Hcl and Int 6,11-dihydro-11-oxo-dibenz[b,e]oxepin-2-acetin acid
  Phosphonium,[3-(dimethylamino)propyl]triphenyl bromide hydrobromide
  6,11-dihydro-11-oxo-dibenz[b,e]oxepin-2-acetin,methyl ester
Palonosetron 5,6,7,8-tetrahydro-1-nephthalenecarboxylic acid
Paroxetine 4,(-)trans-4R-(4-fluorophenyl)-3S-hydroxymethyl-1-methylpiperidine
  (+/-)trans-4R-(4-fluorophenyl)-3S-hydroxymethyl-1-methylpiperidine
  (+/-)trans-3-ethoxy carbonyl-4-(4-flurophenyl)-N-methyl piperidine-2,6-dinone
Perindopril  (2S,3As,7As)-octahydroindole-2-carboxylic acid 
  N-[(S)-1-carbethoxybutyl]-(S)-alanine 
Pregabalin 3-(carbamoylmethyl)-5-methyl hexamoic acid
Ramipril and Int (s,s)-2-azabicyclo [3,3,0] octane-3-carborylic acid benzyl ester hydrochloride 
  (s,s,s)-2-azabicyclo [3,3,0] octane-3-carborylic acid benzyl ester hydrochloride 
Rimonabant Intermediate 5-(4-chlorophenyl-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxylic acid
Rosuvastatin Calcium & Z7,Z8,R3 Z-7 : 4-(4- Fluorophenyl)-6-isopropyl-2-[ (N- methyl-N-methylsulfonyl)amino]pyrimidine-5-yl-methonol
SMIA Sin-Methoxyimino Furanyl Acetic Acid Ammonium Salt
TAA 1,2,3,4-Tetrazolyl-1- Acetic Acid
Tamsulosin  R-(-)-5-(2-Amino-propyl)-2-methoxy-benzenesulfonamide 
  2-(2-Ethoxyphenoxy)bromide ethane 
Ziprasidone 5-Chloroacetyl-6-Chloro-1,3-Dihydro-2-H Indole-2-One 




Intermediates API
2-[3-(Cyano-dimethyl-methyl)-5-methyl-phenyl]-2-methyl-propionitrile  Anastrazole & int
2-methoxy-4-amino-5-ethyl sulfonyl benzoic acid Amisulpride and int.
ATS-5 : (R)-4-cyano-3-hydroxybutyric acid ethyl ester Atorvastatin & ATS-5 ATS-8 ATS -9 M 4 L 1
ATS-8 : (4R,Cis)-1,1-dimethylethyl-cyanomethyl-2,2- dimethyl-1,3-dioxane-4-acetate Atorvastatin & ATS-5 ATS-8 ATS -9 M 4 L 2
Trans-4-chlorophenyl-1-cyclohexane carboxylicacid Atovaquone
(3s,4r)-4-acetoxy-3-[(r)-1-(tert-butyldimethylsilyloxy)ethyl]azetidin-2-1 4-AA
N-[4-Cyano-3-(trifluoromethyl)phenyl]-3-[(4-fluorophenyl)thio]-2-hydroxy-2-methylpropionamide Bicalutamide and int
N-( Triphenylmethyl) ¨C 5-( 4'-bromomethylbiphenyl-2yl) tetrazole Candesartan Cilexetil 
5-(4-Chlorobutyl)-1-Cyclohexyl-1H-Tetrazole Cilostazole 
6-Hydroxy-3,4-dihydro-2(1H)-quinolinone Cilostazole 
2-Thiophene Ethanol  Clopidogrel 
(+)-Methyl-alpha-(2-Thienylethamino) (2-Chlorophenyl) AcetateHydrochloride  Clopidogrel 
N-[(2-Thienyl)ethyl]-(2s)-2-chloro-phenyl Glycine methyl ester  Clopidogrel 
1, 2a -Methylene-6-didehydro -17a -acetoxy Progesterone Cyproterone Acetate
1-Chloromethyl-6-chloro-6-dehydro -17a -acetoxy Progesterone Cyproterone Acetate
2,3-cyclopenteno pyridine CPP
 5,6-Dimethoxy-1-Indanone  Donepezil 
N-Benzyl Piperidine-4-Carboxaldehyde  Donepezil 
2-Bromethyl 1,3 dioxolane Doxofylline and Int.
Ethyl(Z)-2-(2-Aminothiazole-4-yl)-2-Methoxyimino Acetate EHATA
Androsta-1,4-dien-3-one,17-hydoxy-6-methylene(17,β) Exemestane
Androsta-4-ene-3,17-dione,6-methylene(17,β) Exemestane
Ally(1R,2R,5R,6S)-6(1-tert-butyldimethyl siloxyethyl)-2 Faropenem and Int
2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dibenzoate Gemcitabine &int
2-Deoxy-2,2-difluoro pentofuranos-1-ulose-3,5-dibenzoate Gemcitabine &int
2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dicinnamate-1-methane sulfonate Gemcitabine &int
2-Deoxy-2,2-difluoro-D-ribofuranose-3,5-dicinnamate Gemcitabine &int
3-(N-methylpentylamino)propionic acid hydrochloride Ibandronate Sodium
N4-(2-Methylpropyl-3,4-Quinolinediamin Imiquimod and int
1-(1-(s)-(3-(2-(7-chloro-2-qionolinyl)-ethenyl-phenyl)-3-hydroxy-propyl)phenyl)-2-propanol Montelukast sodium
(Z)-2-(tert-methoxycarbonyl methoxyimino)-2-(2-aminothiazol-4-yl) acetic acid MICA ACID
S-2-benzothiazolyl (Z)-2-(2-aminothiazol-4-yl)-2-methoxycarbonylmethoxyiminothio acetate MICA ESTER
4-Amino-2-Methyl-10H-Thieno[2,3-b][1,5]Benxodiazepine Hcl  Olanzapine 
4-chloromethyl-5-methyl-1,3-Dioxol-2-one (DMDO-CL) Olmesartan & int
Trityl Olmesartan Medoxomil Olmesartan & int
6,11-dihydro-11-oxo-dibenz[b,e]oxepin-2-acetin acid Olopatadine Hcl and Int
Phosphonium,[3-(dimethylamino)propyl]triphenyl bromide hydrobromide Olopatadine Hcl and Int
6,11-dihydro-11-oxo-dibenz[b,e]oxepin-2-acetin,methyl ester Olopatadine Hcl and Int
5,6,7,8-tetrahydro-1-nephthalenecarboxylic acid Palonosetron
4,(-)trans-4R-(4-fluorophenyl)-3S-hydroxymethyl-1-methylpiperidine Paroxetine
(+/-)trans-4R-(4-fluorophenyl)-3S-hydroxymethyl-1-methylpiperidine Paroxetine
(+/-)trans-3-ethoxy carbonyl-4-(4-flurophenyl)-N-methyl piperidine-2,6-dinone Paroxetine
(2S,3As,7As)-octahydroindole-2-carboxylic acid  Perindopril 
N-[(S)-1-carbethoxybutyl]-(S)-alanine  Perindopril 
3-(carbamoylmethyl)-5-methyl hexamoic acid Pregabalin
(s,s)-2-azabicyclo [3,3,0] octane-3-carborylic acid benzyl ester hydrochloride  Ramipril and Int
(s,s,s)-2-azabicyclo [3,3,0] octane-3-carborylic acid benzyl ester hydrochloride  Ramipril and Int
5-(4-chlorophenyl-1-(2,4-dichlorophenyl)-4-methylpyrazole-3-carboxylic acid Rimonabant Intermediate
Z-7 : 4-(4- Fluorophenyl)-6-isopropyl-2-[ (N- methyl-N-methylsulfonyl)amino]pyrimidine-5-yl-methonol Rosuvastatin Calcium & Z7,Z8,R3
Sin-Methoxyimino Furanyl Acetic Acid Ammonium Salt SMIA
1,2,3,4-Tetrazolyl-1- Acetic Acid TAA
R-(-)-5-(2-Amino-propyl)-2-methoxy-benzenesulfonamide  Tamsulosin 
2-(2-Ethoxyphenoxy)bromide ethane  Tamsulosin 
5-Chloroacetyl-6-Chloro-1,3-Dihydro-2-H Indole-2-One  Ziprasidone



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